Succinylcholine: Contraindications

Succinylcholine is structurally related to acetylcholine and produces muscle relaxation by first activating muscle fibres, then preventing a further response. As a result, muscle fasciculation is seen in many patients soon after succinylcholine administration. Succinylcholine has a short duration of action as it is metabolized in the plasma by pseudocholinesterase. There are several contraindications to the use of succinylcholine.

Remember that these conditions may also be triggered by using succinylcholine for the first time.

Denervation injury

The initial depolarization, caused by succinylcholine, is reversed by a repolarization that involves potassium moving down its concentration gradient into the extracellular environment. This usually results in a 0.5 mM rise in the plasma concentration of potassium, which is of little clinical significance.
However, where there are extrajunctional receptors, as is seen after denervation injury, the efflux of potassium is much greater and may cause a clinically significant rise in potassium concentration, resulting in ventricular fibrillation followed by asystole.

Eye injury

Contraction of the extra-ocular muscles following the use of succinylcholine result in a significant rise in intraocular pressure so that the contents of the eyeball may be compromised where there is an open eye injury.